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ALLWOOD, Daniel, BLAKEMORE, David C., BROWN, Alan D. and LEY, Steven V. (2014). Metal-free coupling of saturated heterocyclic sulfonylhydrazones with boronic acids. The Journal of Organic Chemistry, 79 (1), 328-338.
Full text not available from this repository.Abstract
The coupling of aromatic moieties with saturated heterocyclic partners is currently an area of significant interest for the pharmaceutical industry. Herein, we present a procedure for the metal-free coupling of 4-, 5-, and 6-membered saturated heterocyclic p-methoxyphenyl (PMP) sulfonylhydrazones with aryl and heteroaromatic boronic acids. This procedure enables a simple, two-step synthesis of a range of functionalized sp2−sp3 linked bicyclic building blocks, including oxetanes, piperidines, and azetidines, from their parent ketones. ■ INTRODUCTION
| Item Type: | Article |
|---|---|
| Research Institute, Centre or Group - Does NOT include content added after October 2018: | Biomedical Research Centre |
| Identification Number: | https://doi.org/10.1021/jo402526z |
| Page Range: | 328-338 |
| Depositing User: | Users 3084 not found. |
| Date Deposited: | 13 Aug 2015 09:03 |
| Last Modified: | 17 Mar 2021 19:31 |
| URI: | https://shura.shu.ac.uk/id/eprint/10758 |
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